The efficacy of folic acid (FA) and folinic acid (FNA) reducing methotrexate (MTX) side effects in rheumatoid arthritis (RA)

Article type
Authors
Ortiz Z, Shea B, Suarez AM, Moher D, Wells G, Tugwell P
Abstract
Introduction: MTX is an antimetabolite used in the treatment of RA and is considered to be the second-line drug of first choice. MTX's side effects occur in about 60% of patients. Some side effects mimic complicated folate deficiency. Several studies have been conducted to determine if folate supplementation has a beneficial effect reducing MTX side-effects, without altering its efficacy, but the answer remains uncertain.

Objective: To determine the efficacy of FA and FNA to reduce gastrointestinal and haematologic side effects of low-dose MTX in patients with RA, and whether or not folate supplementation alters MTX efficacy.

Methods: Using the Cochrane Musculoskeletal Group search strategy, we selected all double-blind, placebo-controlled randomised clinical trials in patients who fulfilled the American Rheumatism Association's criteria for RA, older than 18 years, treated with low dose MTX (less than 20 mg/week) concurrently with folate supplementation. The outcomes were the reduction of GI and/or haematologic side effects, and the efficacy of MTX in patients who received folate supplementation. Treatment effect was calculated using a fixed effect model (Peto). Sensitivity analysis was done to compare the results with different doses and different quality of trials.

Results: Six RCTs fulfilled the inclusion criteria. Haematologic side effects could not be analysed. A significant reduction in the odds of GI side effects of 68% was shown. Considering trials that use a dose of FA or FNA less than 10mg/week, there was a significant reduction in GI side effects of 75%.

Discussion: Folate supplementation has a protective effect, reducing MTX related GI side effects, without affecting MTX efficacy. No evidence has shown that FA or FNA is the most effective.